| 產品名稱 | ARN 272 |
| 產品貨號 | Axon 2941 CAS [488793-85-7] MF C27H20N4O2MW 432.47 Purity: 98% Soluble in DMSO Recently added |
| 產品價格 | 現貨詢價,電話:010-67529703 |
| 產品規格 | |
| 產品品牌 | axonmedchem |
| 產品概述 | |
| 產品詳情 |
ARN 272Axon 2941 CAS [488793-85-7] MF C27H20N4O2
Recently added
DescriptionARN 272 is a selective competitive antagonist of the interaction of anandamide with FAAH-like anandamide transporter (IC50 value of 1.8 μM). Moreover, ARN 272 prevents anandamide internalization in vitro, interrupts anandamide deactivation in vivo, and exerts profound analgesic effects in rodent models of nociceptive and inflammatory pain, which are mediated by CB1 cannabinoid receptors. KEYWORDS: ARN 272 | supplier | FLAT inhibitor | ARN272 | ARN-272 | CAS [488793-85-7] | Fatty acid (Amides) | FLAT | Inhibitor | Proteins | FAAH-1
Selective inhibitor of FAAH-like anandamide transporter (FLAT)
Chemical name4-(4-(4-Hydroxyphenyl)phthalazin-1-ylamino)-N-phenylbenzamide Parent CAS No.[488793-85-7] |
| 產品資料 |