| 產品名稱 | KDM5 inhibitor compound 48 |
| 產品貨號 | Axon 2809 CAS [1628210-26-3] MF C17H20N6OMW 324.38 Purity: 99% Soluble in DMSO Description Potent, selective and orally bioavailable KDM5 inhibitor (IC50 value of 15.1 nM for KDM5A) with improved cell potency (EC50 value of 0.34 μM, H3K4Me3 level in PC9 cells). Chemical probe suitable for studying KDM5 biological functions in vivo. KEYWORDS: KDM5 inhibitor compound 48 | supplier | KDM5 inhibitor | CAS [1628210-26-3] | Histone demethylase | Inhibitor | Enzymes | Orally bioavailable | PC9 |
| 產品價格 | 現貨詢價,電話:010-67529703 |
| 產品規格 | |
| 產品品牌 | axonmedchem |
| 產品概述 | |
| 產品詳情 |
KDM5 inhibitor compound 48Axon 2809 CAS [1628210-26-3] MF C17H20N6O
DescriptionPotent, selective and orally bioavailable KDM5 inhibitor (IC50 value of 15.1 nM for KDM5A) with improved cell potency (EC50 value of 0.34 μM, H3K4Me3 level in PC9 cells). Chemical probe suitable for studying KDM5 biological functions in vivo. KEYWORDS: KDM5 inhibitor compound 48 | supplier | KDM5 inhibitor | CAS [1628210-26-3] | Histone demethylase | Inhibitor | Enzymes | Orally bioavailable | PC9
Selective and orally bioavailable KDM5 inhibitor
Chemical name5-(1-tert-Butyl-1H-pyrazol-4-yl)-6-isopropyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile Parent CAS No.[1628210-26-3] |
| 產品資料 |